99% byera cyane CAS 7361-61-7
Gukoresha Xylazine
X.Analogogue ya clonidine, ni agonist kurwego rwa α2 rwakirwa rya adrenergic.Xylazine aherutse kwigaragaza nk'ibiyobyabwenge byo kwidagadura, cyane cyane muri Porto Rico [1].Ubuyobozi bwa xylazine (0.17 mg / kg yuburemere bwumubiri, bugabanijwe kugeza kuri ml-10, ukoresheje 0.9% NaCl) bwateje amasaha agera kuri 2.5 ya analgesia yaho nta ngaruka zigaragara.Umubare munini wa xylazine wateje inyuma yinyuma yinyuma ataxia.Ubuyobozi bwa lidocaine bwateje igihe gisa na analgesia, hamwe na ataxia yinyuma yinyuma (100%).Twanzuye ko xylazine itangwa no gutera inshinge zitera analgesie itekanye, ikora neza mumafarasi [2].
Igikorwa cyibinyabuzima cya Xylazine
Ibisobanuro | X.Analogogue ya clonidine, ni agonist kurwego rwa α2 rwakirwa rya adrenergic.Xylazine aherutse kwigaragaza nk'ibiyobyabwenge byo kwidagadura, cyane cyane muri Porto Rico [1].Ubuyobozi bwa xylazine (0.17 mg / kg yuburemere bwumubiri, bugabanijwe kugeza kuri ml-10, ukoresheje 0.9% NaCl) bwateje amasaha agera kuri 2.5 ya analgesia yaho nta ngaruka zigaragara.Umubare munini wa xylazine wateje inyuma yinyuma yinyuma ataxia.Ubuyobozi bwa lidocaine bwateje igihe gisa na analgesia, hamwe na ataxia yinyuma yinyuma (100%).Twanzuye ko xylazine itangwa no gutera inshinge zitera analgesie itekanye, ikora neza mumafarasi [2]. | ||||||||||||
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Cataloge bifitanye isano | Inzira Yerekana Ibimenyetso >> GPCR / G Poroteyine >> Kwakira Adrenergic Ibice byubushakashatsi >> Indwara zifata ubwonko | ||||||||||||
Umuti | Muri Vitro: MM 10 muri DMSO | ||||||||||||
Gukemura |
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Ububiko | Nyamuneka ubike ibicuruzwa mubihe bisabwa muri Certificat ya Analyse. | ||||||||||||
Kohereza | Ubushyuhe bwicyumba kumugabane wa Amerika;Birashobora gutandukana ahandi | ||||||||||||
URWENYA | CC1 = C (C (C) = CC = C1) NC2 = NCCCS2 | ||||||||||||
Reba | [1].Reyes, JC, n'abandi, Kugaragara kwa xylazine nk'umuti mushya w'ihohoterwa n'ingaruka z’ubuzima mu bakoresha ibiyobyabwenge muri Porto Rico.J Ubuzima bwo mu Mijyi, 2012. 89 (3): p.519-26. [2].Hsu, WH, Xylazine iterwa no kwiheba hamwe na antagonism yayo na alpha adrenergic yo gukumira.J Pharmacol Ikwirakwiza, 1981. 218 (1): p.188-92. | ||||||||||||
Ibijyanye na molekile | Isoprenaline hydrochloride |ICI 118,551 (hydrochloride) |Fenilephrine hydrochloride |Yohimbine hydrochloride |L (-) - Epinephrine |Ivabradine hydrochloride |Prazosin hydrochloride |Clenbuterol hydrochloride |Phentolamine mesilate |guanfacine hydrochloride |pimozide |Sotalol hydrochloride |Carvedilol |Atenolol |Metroprolol irasimburana |
Amakuru yuburozi
Amakuru yuburozi
KUMENYA KIMI
UBUZIMA BWA DATADATA YUBUMWE
|
Synonyme
Rompun |
Xylazinum |
xylazine |
MFCD00057908 |
Xilazina [INN-Espanye] |
EINECS 230-902-1 |
4H-1,3-Thiazin-2-amine, N- (2,6-dimethylphenyl) -5,6-dihydro- |
UNII-2KFG9TP5V8 |
N- (2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine |
Xylazinum [INN-Ikilatini] |
Xylazin |
Xilazina |
(5,6-dihydro-4H- [1,3] thiazin-2-yl) - (2,6-dimethyl-phenyl) -amine |
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