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99% byera cyane CAS 7361-61-7

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    Ibicuruzwa

    5449-12-7

    Izina Rusange Xylazine
    Umubare CAS 7361-61-7 Uburemere bwa molekile 220.334
    Ubucucike 1.2 ± 0.1 g / cm3 Ingingo 334.2 ± 52.0 ° C kuri 760 mmHg
    Inzira ya molekulari C12H16N2S Ingingo yo gushonga 140ºC
    MSDS hfgc

    Igishinwa Amerika

    Flash point 155.9 ± 30.7 ° C.
    Ikimenyetso GHS06
    GHS06
    Ijambo ry'ikimenyetso Akaga

    7361-61-7 (3) 7361-61-7 (2) 7361-61-7 (1) gupakira (7) gupakira (6)

    Gukoresha Xylazine

    X.Analogogue ya clonidine, ni agonist kurwego rwa α2 rwakirwa rya adrenergic.Xylazine aherutse kwigaragaza nk'ibiyobyabwenge byo kwidagadura, cyane cyane muri Porto Rico [1].Ubuyobozi bwa xylazine (0.17 mg / kg yuburemere bwumubiri, bugabanijwe kugeza kuri ml-10, ukoresheje 0.9% NaCl) bwateje amasaha agera kuri 2.5 ya analgesia yaho nta ngaruka zigaragara.Umubare munini wa xylazine wateje inyuma yinyuma yinyuma ataxia.Ubuyobozi bwa lidocaine bwateje igihe gisa na analgesia, hamwe na ataxia yinyuma yinyuma (100%).Twanzuye ko xylazine itangwa no gutera inshinge zitera analgesie itekanye, ikora neza mumafarasi [2].

    Igikorwa cyibinyabuzima cya Xylazine

    Ibisobanuro X.Analogogue ya clonidine, ni agonist kurwego rwa α2 rwakirwa rya adrenergic.Xylazine aherutse kwigaragaza nk'ibiyobyabwenge byo kwidagadura, cyane cyane muri Porto Rico [1].Ubuyobozi bwa xylazine (0.17 mg / kg yuburemere bwumubiri, bugabanijwe kugeza kuri ml-10, ukoresheje 0.9% NaCl) bwateje amasaha agera kuri 2.5 ya analgesia yaho nta ngaruka zigaragara.Umubare munini wa xylazine wateje inyuma yinyuma yinyuma ataxia.Ubuyobozi bwa lidocaine bwateje igihe gisa na analgesia, hamwe na ataxia yinyuma yinyuma (100%).Twanzuye ko xylazine itangwa no gutera inshinge zitera analgesie itekanye, ikora neza mumafarasi [2].
    Cataloge bifitanye isano
    Inzira Yerekana Ibimenyetso >> GPCR / G Poroteyine >> Kwakira Adrenergic
    Ibice byubushakashatsi >> Indwara zifata ubwonko
    Umuti
    Muri Vitro:

    MM 10 muri DMSO

    Gukemura
    1 mM 4.5386 mL 22.6932 mL 45.3865 mL
    5 mM 0,9077 mL 4.5386 mL 9.0773 mL
    10 mM 0.4539 mL 2.2693 mL 4.5386 mL
    Ububiko Nyamuneka ubike ibicuruzwa mubihe bisabwa muri Certificat ya Analyse.
    Kohereza Ubushyuhe bwicyumba kumugabane wa Amerika;Birashobora gutandukana ahandi
    URWENYA CC1 = C (C (C) = CC = C1) NC2 = NCCCS2
    Reba [1].Reyes, JC, n'abandi, Kugaragara kwa xylazine nk'umuti mushya w'ihohoterwa n'ingaruka z’ubuzima mu bakoresha ibiyobyabwenge muri Porto Rico.J Ubuzima bwo mu Mijyi, 2012. 89 (3): p.519-26.

    [2].Hsu, WH, Xylazine iterwa no kwiheba hamwe na antagonism yayo na alpha adrenergic yo gukumira.J Pharmacol Ikwirakwiza, 1981. 218 (1): p.188-92.

    Ibijyanye na molekile Isoprenaline hydrochloride |ICI 118,551 (hydrochloride) |Fenilephrine hydrochloride |Yohimbine hydrochloride |L (-) - Epinephrine |Ivabradine hydrochloride |Prazosin hydrochloride |Clenbuterol hydrochloride |Phentolamine mesilate |guanfacine hydrochloride |pimozide |Sotalol hydrochloride |Carvedilol |Atenolol |Metroprolol irasimburana

    Amakuru yuburozi

    Amakuru yuburozi

    KUMENYA KIMI

    UMUBARE WA RTECS:
    XJ0776300
    IZINA RYA CHIMIQUE:
    4H-1,3-Thiazine, 5,6-dihydro-2- (2,6-xylidino) -
    UMUBARE WO KWIYANDIKISHA:
    7361-61-7
    AMAKURU MASO MASHYA:
    199606
    INGINGO ZA DATA:
    8
    FORMULA MOLECULAR:
    C12-H16-N2-S
    UBUREMERE BWA MOLECULAR:
    220.36
    UMWANZURO WITONDE:
    T6N CS AUTJ BMR B1 F1

    UBUZIMA BWA DATA

    DATA YUBUMWE

    UBWOKO BW'IKIZAMINI:
    TDLo - Igipimo gito cyatangajwe
    INZIRA YO KUGARAGAZA:
    Umunwa
    UMWIHARIKO YAKurikiranwe:
    Umuntu - umugore
    DOSE / DURATION:
    8 mg / kg
    INGARUKA Z'UBURYO:
    Imyitwarire - somnolence (ibikorwa rusange byihebye) Imyitwarire - impinduka mubikorwa bya moteri (assay yihariye) Cardiac - igipimo cya pulse
    BIKORWA:
    CTOXAO Uburozi bwa Clinical.(New York, NY) V.1-18, 1968-81.Kumakuru yamamaza, reba JTCTDW.Igitabo (ikibazo) / urupapuro / umwaka: 18,663,1981
    UBWOKO BW'IKIZAMINI:
    TDLo - Igipimo gito cyatangajwe
    INZIRA YO KUGARAGAZA:
    Intramuscular
    UMWIHARIKO YAKurikiranwe:
    Umuntu - umugore
    DOSE / DURATION:
    734 ug / kg
    INGARUKA Z'UBURYO:
    Inzego Zibyumva hamwe na Sens idasanzwe (Ijisho) - miose (impagarike yumunyeshuri) Umutima - igipimo cyumuvuduko wamaraso - BP kugabanuka ntabwo irangwa mubice byigenga
    BIKORWA:
    AJEMEN Ikinyamakuru cyo muri Amerika cyubuvuzi bwihutirwa.(WB Saunders, Philadelphia, PA) V.1- 1983- Igitabo (nomero) / urupapuro / umwaka: 4,222.1986
    UBWOKO BW'IKIZAMINI:
    TDLo - Igipimo gito cyatangajwe
    INZIRA YO KUGARAGAZA:
    Intramuscular
    UMWIHARIKO YAKurikiranwe:
    Umuntu - umugore
    DOSE / DURATION:
    22 mg / kg
    INGARUKA Z'UBURYO:
    Imyitwarire - somnolence (ibikorwa byihebye muri rusange) Umutima - igipimo cyimisemburo Ibihaha, Thorax, cyangwa Guhumeka - kubyimba neza
    BIKORWA:
    AJEMEN Ikinyamakuru cyo muri Amerika cyubuvuzi bwihutirwa.(WB Saunders, Philadelphia, PA) V.1- 1983- Igitabo (nomero) / urupapuro / umwaka: 4,222.1986
    UBWOKO BW'IKIZAMINI:
    LD50 - Igipimo cyica, 50 ku ijana byica
    INZIRA YO KUGARAGAZA:
    Umunwa
    UMWIHARIKO YAKurikiranwe:
    Imbeba - imbeba
    DOSE / DURATION:
    130 mg / kg
    INGARUKA Z'UBURYO:
    Ibisobanuro byingaruka zuburozi ntabwo byatangajwe usibye agaciro kica
    BIKORWA:
    DTTIAF Deutsche Tieraerztliche Wochenschrift.(Hanover, Fed. Depite Ger.) V.1-77, 1893-1970.Igitabo (ikibazo) / urupapuro / umwaka: 75.565.1968
    UBWOKO BW'IKIZAMINI:
    LD50 - Igipimo cyica, 50 ku ijana byica
    INZIRA YO KUGARAGAZA:
    Umunwa
    UMWIHARIKO YAKurikiranwe:
    Imbeba - imbeba
    DOSE / DURATION:
    240 mg / kg
    INGARUKA Z'UBURYO:
    Ibisobanuro byingaruka zuburozi ntabwo byatangajwe usibye agaciro kica
    BIKORWA:
    DTTIAF Deutsche Tieraerztliche Wochenschrift.(Hanover, Fed. Depite Ger.) V.1-77, 1893-1970.Igitabo (ikibazo) / urupapuro / umwaka: 75.565.1968
    UBWOKO BW'IKIZAMINI:
    LD50 - Igipimo cyica, 50 ku ijana byica
    INZIRA YO KUGARAGAZA:
    Subcutaneous
    UMWIHARIKO YAKurikiranwe:
    Imbeba - imbeba
    DOSE / DURATION:
    121 mg / kg
    INGARUKA Z'UBURYO:
    Ibisobanuro byingaruka zuburozi ntabwo byatangajwe usibye agaciro kica
    BIKORWA:
    DTTIAF Deutsche Tieraerztliche Wochenschrift.(Hanover, Fed. Depite Ger.) V.1-77, 1893-1970.Igitabo (ikibazo) / urupapuro / umwaka: 75.565.1968
    UBWOKO BW'IKIZAMINI:
    LD50 - Igipimo cyica, 50 ku ijana byica
    INZIRA YO KUGARAGAZA:
    Imitsi
    UMWIHARIKO YAKurikiranwe:
    Imbeba - imbeba
    DOSE / DURATION:
    18 mg / kg
    INGARUKA Z'UBURYO:
    Ibisobanuro byingaruka zuburozi ntabwo byatangajwe usibye agaciro kica
    BIKORWA:
    CSLNX * Ingabo z’Amerika Intwaro Ubushakashatsi & Iterambere, Ubuyobozi bwa Laboratwari, Laboratoire ya NIOSH.. - E0475 No.

    Synonyme

    Rompun
    Xylazinum
    xylazine
    MFCD00057908
    Xilazina [INN-Espanye]
    EINECS 230-902-1
    4H-1,3-Thiazin-2-amine, N- (2,6-dimethylphenyl) -5,6-dihydro-
    UNII-2KFG9TP5V8
    N- (2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine
    Xylazinum [INN-Ikilatini]
    Xylazin
    Xilazina
    (5,6-dihydro-4H- [1,3] thiazin-2-yl) - (2,6-dimethyl-phenyl) -amine

    Isosiyete yacu

    Wuhan Xiju Biotechnology Co, Ltd. ni uruganda rukora umwuga wo gukora imiti mvaruganda.Isosiyete ifite itsinda ryigenga ryubushakashatsi niterambere, rishobora gukora ubushakashatsi no guteza imbere ibikoresho byose byubuvuzi, hamwe nigiciro gito, cyiza kandi na serivisi yo mucyiciro cya mbere!

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